Neurokinin Receptor Inhibitors

NK1R

NK2R

NK3R

Neurokinin Receptor Inhibitors, Agonists, Antagonists & Modulators

Product Name	NK1R	NK2R	NK3R	Purity
Substance P	NK1R			99.82%
Senktide	NK1R, EC₅₀: 35 nM		NK3R, EC₅₀: 0.5-3 nM	99.85%
Fezolinetant			NK3R	99.19%
Senktide TFA	NK1R, EC₅₀: 35 μM		NK3R, EC₅₀: 0.5-3 nM
Rolapitant	monkey NK1, Ki: 2.5 nM rat NK1, Ki: 78.6 nM rabbit NK1, Ki: 31.7 nM gerbil NK1, Ki: 0.13 nM guinea pig NK1, Ki: 0.72 nM human NK1, Ki: 0.66 nM mouse NK1, Ki: 60.4 nM			99.89%
EB1002		NK2R		99.91%
Saredutant		NK2R		98.09%
SB-222200			NK3R	99.85%
L-732138	NK1R, IC₅₀: 2.3 nM			≥99.9%
N-Acetyl-L-tryptophan	NK1R			99.38%
Talnetant			NK3R	99.48%
Orvepitant maleate	NK1R, pKi: 10.2			99.99%
L-733060 hydrochloride	NK1R			99.30%
Osanetant			NK3R	98.19%
Maropitant	NK1R			99.52%
Casopitant mesylate	NK1R			99.83%
Substance P TFA	NK1R
Pavinetant			NK3R	99.83%
Eprazinone dihydrochloride	NK1R			99.05%
Vofopitant dihydrochloride	NK1R			99.56%
Vapreotide	NK1R			99.87%
Spantide II	NK1R			98.01%
Eledoisin		NK2R	NK3R	99.05%
Hemokinin 1 (mouse)	NK1R			99.49%
[Lys5,MeLeu9,Nle10]Neurokinin A(4-10)		NK2R		99.83%
Hemokinin 1, human	NK1R	NK2R	NK3R	98.11%
Biotin-Substance P	NK1R			99.91%
GR 159897		hNK2, pKi: 9.51 (CHO cell) NK2R, pKi: 10 (Rat colon membrane)		99.60%
Spantide I	NK1R, Ki: 230 nM	NK2R, Ki: 8150 nM		99.72%
MEN 10207	NK1R, pA2: 5.2	Tachykinin NK₂ Receptor, pA2: 7.9	NK3R, pA2: 4.9	99.69%
Rolapitant hydrochloride hydrate	monkey NK1, Ki: 2.5 nM rat NK1, Ki: 78.6 nM rabbit NK1, Ki: 31.7 nM gerbil NK1, Ki: 0.13 nM guinea pig NK1, Ki: 0.72 nM human NK1, Ki: 0.66 nM mouse NK1, Ki: 60.4 nM			98.25%
[MePhe7]-Neurokinin B			NK3R, IC₅₀: 3 nM	98.87%
Fosnetupitant chloride monohydrochloride	hNK1, pKi: 9.5		hNK3, pKi: 6.1	99.70%
Vapreotide acetate	NK1R			99.85%
γ-Neuropeptide (rabbit)		NK2R		99.99%
L-760735	hNK1, IC₅₀: 0.19 nM			≥99.0%
SB 218795		hNK2, Ki: 1220 nM	hNK3, Ki: 13 nM	99.86%
Nolpitantium	NK1R
GR 87389		NK2R
Hemokinin 1, human TFA	NK1R	NK2R	NK3R
(D-Arg1,D-Pro2,D-Phe7,D-His9)-Substance P	NK1R
GR 94800 TFA		NK2R
[D-Trp2,7,9] Substance P	NK1R, Ki: 1 μM	NK2R, Ki: 1.3 μM	NK3R, Ki: ~9 μM
[Pro9]-Substance P	NK1R, EC₅₀: 0.93 nM
Scyliorhinin I	rat NK1, Ki: 0.9 nM	guinea pig NK-2, Ki: 2 nM
Rolapitant hydrochloride	monkey NK1, Ki: 2.5 rat NK1, Ki: 78.6 rabbit NK1, Ki: 31.7 gerbil NK1, Ki: 0.13 guinea pig NK1, Ki: 0.72 human NK1, Ki: 0.66 mouse NK1, Ki: 60.4
Acetylaszonalenin	NK1R
Neurokinin Receptor (393-407), rat	NK1R
SSR 146977			NK3R
L-741671	hNK1, Ki: 0.03 nM
(Trp7,β-Ala8)-Neurokinin A (4-10)			NK3R
CP 122721 hydrochloride	human NK1, pIC₅₀: 9.8
SDZ NKT 343	hNK1, IC₅₀: 0.62 nM	hNK2, Ki: 0.52 μM	hNK3, Ki: 3.4 μM
Imnopitant	NK1R
Phyllomedusin	NK1R
CS-003 Free base	NK1R, Ki: 2.3 nM	NK2R, Ki: 0.54 nM
ASN-1377642	NK1R, Ki: 251 nM
Maropitant citrate	NK1R
Fosrolapitant	NK1R
ZM 253270		Hamster Bladder NK-2, Ki: 2 nM
YM-49598 iodide	NK1R
Befetupitant	NK1R
Vestipitant	hNK1, pKi: 9.4
Talnetant hydrochloride			NK3R
Physalaemin	NK1R

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