1. Signaling Pathways
  2. GPCR/G Protein
    Neuronal Signaling
  3. Neurokinin Receptor
  4. Neurokinin Receptor Inhibitors

Neurokinin Receptor Inhibitors

NK1R

NK2R

NK3R

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

Neurokinin Receptor Inhibitors, Agonists, Antagonists & Modulators
Product Name NK1R NK2R NK3R Purity
Substance P
NK1R
    99.82%
Senktide
NK1R, EC50: 35 nM
 
NK3R, EC50: 0.5-3 nM
99.85%
Fezolinetant    
NK3R
99.19%
Senktide TFA
NK1R, EC50: 35 μM
 
NK3R, EC50: 0.5-3 nM
Rolapitant
monkey NK1, Ki: 2.5 nM
rat NK1, Ki: 78.6 nM
rabbit NK1, Ki: 31.7 nM
gerbil NK1, Ki: 0.13 nM
guinea pig NK1, Ki: 0.72 nM
human NK1, Ki: 0.66 nM
mouse NK1, Ki: 60.4 nM
    99.89%
EB1002  
NK2R
  99.91%
Saredutant  
NK2R
  98.09%
SB-222200    
NK3R
99.85%
L-732138
NK1R, IC50: 2.3 nM
    ≥99.9%
N-Acetyl-L-tryptophan
NK1R
    99.38%
Talnetant    
NK3R
99.48%
Orvepitant maleate
NK1R, pKi: 10.2
    99.99%
L-733060 hydrochloride
NK1R
    99.30%
Osanetant    
NK3R
98.19%
Maropitant
NK1R
    99.52%
Casopitant mesylate
NK1R
    99.83%
Substance P TFA
NK1R
   
Pavinetant    
NK3R
99.83%
Eprazinone dihydrochloride
NK1R
    99.05%
Vofopitant dihydrochloride
NK1R
    99.56%
Vapreotide
NK1R
    99.87%
Spantide II
NK1R
    98.01%
Eledoisin  
NK2R
NK3R
99.05%
Hemokinin 1 (mouse)
NK1R
    99.49%
[Lys5,MeLeu9,Nle10]Neurokinin A(4-10)  
NK2R
  99.83%
Hemokinin 1, human
NK1R
NK2R
NK3R
98.11%
Biotin-Substance P
NK1R
    99.91%
GR 159897  
hNK2, pKi: 9.51 (CHO cell)
NK2R, pKi: 10 (Rat colon membrane)
  99.60%
Spantide I
NK1R, Ki: 230 nM
NK2R, Ki: 8150 nM
  99.72%
MEN 10207
NK1R, pA2: 5.2
Tachykinin NK2 Receptor, pA2: 7.9
NK3R, pA2: 4.9
99.69%
Rolapitant hydrochloride hydrate
monkey NK1, Ki: 2.5 nM
rat NK1, Ki: 78.6 nM
rabbit NK1, Ki: 31.7 nM
gerbil NK1, Ki: 0.13 nM
guinea pig NK1, Ki: 0.72 nM
human NK1, Ki: 0.66 nM
mouse NK1, Ki: 60.4 nM
    98.25%
[MePhe7]-Neurokinin B    
NK3R, IC50: 3 nM
98.87%
Fosnetupitant chloride monohydrochloride
hNK1, pKi: 9.5
 
hNK3, pKi: 6.1
99.70%
Vapreotide acetate
NK1R
    99.85%
γ-Neuropeptide (rabbit)  
NK2R
  99.99%
L-760735
hNK1, IC50: 0.19 nM
    ≥99.0%
SB 218795  
hNK2, Ki: 1220 nM
hNK3, Ki: 13 nM
99.86%
Nolpitantium
NK1R
   
GR 87389  
NK2R
 
Hemokinin 1, human TFA
NK1R
NK2R
NK3R
(D-Arg1,D-Pro2,D-Phe7,D-His9)-Substance P
NK1R
   
GR 94800 TFA  
NK2R
 
[D-Trp2,7,9] Substance P
NK1R, Ki: 1 μM
NK2R, Ki: 1.3 μM
NK3R, Ki: ~9 μM
[Pro9]-Substance P
NK1R, EC50: 0.93 nM
   
Scyliorhinin I
rat NK1, Ki: 0.9 nM
guinea pig NK-2, Ki: 2 nM
 
Rolapitant hydrochloride
monkey NK1, Ki: 2.5
rat NK1, Ki: 78.6
rabbit NK1, Ki: 31.7
gerbil NK1, Ki: 0.13
guinea pig NK1, Ki: 0.72
human NK1, Ki: 0.66
mouse NK1, Ki: 60.4
   
Acetylaszonalenin
NK1R
   
Neurokinin Receptor (393-407), rat
NK1R
   
SSR 146977    
NK3R
L-741671
hNK1, Ki: 0.03 nM
   
(Trp7,β-Ala8)-Neurokinin A (4-10)    
NK3R
CP 122721 hydrochloride
human NK1, pIC50: 9.8
   
SDZ NKT 343
hNK1, IC50: 0.62 nM
hNK2, Ki: 0.52 μM
hNK3, Ki: 3.4 μM
Imnopitant
NK1R
   
Phyllomedusin
NK1R
   
CS-003 Free base
NK1R, Ki: 2.3 nM
NK2R, Ki: 0.54 nM
 
ASN-1377642
NK1R, Ki: 251 nM
   
Maropitant citrate
NK1R
   
Fosrolapitant
NK1R
   
ZM 253270  
Hamster Bladder NK-2, Ki: 2 nM
 
YM-49598 iodide
NK1R
   
Befetupitant
NK1R
   
Vestipitant
hNK1, pKi: 9.4
   
Talnetant hydrochloride    
NK3R
Physalaemin
NK1R